- Article
- Afatinib
- Product Number
- S1011-1G
- Supplier
- Selleck Chemicals
- Size
- 1 g
- Description
- Afatinib inhibits EGFR/ErbB irreversibly in vitro with IC50 of 0.5, 0.4, 10, 14, 1 nM for EGFRwt, EGFR L858R , EGFR L858R/T790M ErbB2 (HER2) and ErbB4 (HER4), respectively. Afatinib induces autophagy.
- Category
- Proteins, Peptides and Small Molecules
- Product Group
- Inhibitors & Activators
- CAS Number
- 850140-72-6
- Formulation
- C24H25ClFN5O3
- Shipping Temperature
- BLUE ICE
- Supplier URL
- Visit supplier product page